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Neurochemicals and neurosteroids modulations of 4-(2-chloro-4-fluorobenzyl)-3-(2-thienyl)-1,2,4-oxadiazol-5(4H)-one on the pentylenetetrazole-induced epileptic seizure in the zebrafish model
Author
Seong Soon Kim, Hyemin Kan, Kyu-Seok Hwang, Jung Yoon Yang, Yuji Son, Dae-Seop Shin, Byung Hoi Lee, Se Hwan Ahn, Jin Hee Ahn, Sung-Hee Cho*, Myung Ae Bae*
Year
2021
Source
Int. J. Mol. Sci. 2021, 22, 1285
Design, Synthesis, and Biological Evaluation of New Peripheral 5HT2A Antagonists for Nonalcoholic Fatty Liver Disease
Author
Minhee Kim, Inseon Hwang, Haushabhau S. Pagire, Suvarna H Pagire, Wonsuk Choi, Won Gun Choi, Jihyeon Yoon, Won Mi Lee, Jin Sook Song, Eun Kyung Yoo, Seungmi Lee, Mijin Kim, Myung Ae Bae, Dooseop Kim, Heejong Lee, Eun-Young Lee, Jae-Han Jeon, In Kyu Lee, Hail Kim*, Jin Hee Ahn*
Year
2020
Source
J. Med. Chem. 2020, 63, 4171-4182
Identification of novel anti-melanogenic agents using a zebrafish model
Author
Se Hwan Ahn, Kyu-Seok Hwang, Dae-Seop Shin, Seong Soon Kim, Jung Yoon Yang, Myung Ae Bae*, Jin Hee Ahn*
Year
2020
Source
Bioorg. & Med. Chem. Lett. 2020, 30,127201
Optimization of cyclic sulfamide derivatives as 11beta-hydroxysteroid dehydrogenase 1 inhibitors for the potential treatment of ischemic brain injury
Author
Jeong Hyun Lee, Ju Hwan Bok, Sung Bum Park, Haushabhau S. Pagire, Yoon-Ju Na, Won Hoon Jung, Jin Sook Song, Nam Sook Kang, Ho Won Seo, Byung Ho Lee, Ki Young Kim*, Jin Hee Ahn*
Year
2020
Source
Bioorg. & Med. Chem. Lett. 2020, 30, 126787
Multimodal imaging probe development for pancreatic β-cells: from fluorescence to PET
Author
Nam-Young Kang, Jung Yeol Lee, Sang Hee Lee, In Ho Song, Yong Hwa Hwang, Min Jun Kim,Wut Hmone Phue, Bikram Keshari Agrawalla, Si Yan Diana Wan, Janise Lalic, Sung-Jin Park, Jong-Jin Kim, Haw-Young Kwon, So Hee Im, Myung Ae Bae, Jin Hee Ahn, Chang Siang Lim, Adrian Kee Keong Teo, Sunyou Park, Sang Eun Kim, Byung Chul Leel, Dong Yun Lee, Young-Tae Chang *
Year
2020
Source
J. Am. Chem. Soc. 2020, 147, 3430-3439
TMBIM6/BI-1 contributes to cancer progression through assembly with mTORC2 and AKT activation
Author
Hyun-Kyoung Kim, Kashi Raj Bhattarai, Raghu Patil Junjappa, Jin Hee Ahn, Suvarna H. Pagire, Hyun Ju Yoo, Jaeseok Han, Duckgue Lee, Kyung-Woon Kim, Hyung-Ryong Kim, Han-Jung Chae*
Year
2020
Source
Nature Communications 2020, 11, 4012
Structural basis for the inhibition of PDK2 by novel ATP- and lipoylbinding site targeting compounds
Author
Jihoon Kang, Haushabhau S. Pagire, Donguk Kang, Yo Han Song, In Kyu Lee, Kang Taek Lee, Chin-Ju Park, Jin Hee Ahn, Jungwook Kim*
Year
2020
Source
Biochemical and Biophysical Research Communications 2020, 527, 778-784
Efficacy and pharmacokinetics evaluation of 4-(2-chloro-4-fluorobenzyl)-3-(2-thienyl)-1,2,4-oxadiazol-5(4H)-one (GM-90432) as an anti-seizure agent
Author
Kyu-Seok Hwang, Hyemin Kan, Seong Soon Kim, Jin Sil Chae, Jung Yoon Yang, Dae-Seop Shin, Se Hwan Ahn, Jin Hee Ahn, Jin-Hwa Cho, Il-Sung Jang, Cheol-Hee Kim, and Myung Ae Bae*
Year
2020
Source
Neurochemistry International 2020, 141, 104870
Potent Small-molecule Inhibitors Targeting Acetylated Microtubules as Anticancer Agents against Triple-negative Breast Cancer
Author
Ahreum Kwon, Gwi Bin Lee, Taein Park, Jung Hoon Lee, Panseon Ko, Eunae You, Jin Hee Ahn, Soo Hyun Eom, Sangmyung Rhee*, and Woo Keun Song*
Year
2020
Source
Biomedicine 2020 8, 338
A Novel Selective 11-HSD1 Inhibitor, (E)-4-(2-(6-(2,6-Dichloro-4-(Trifluoromethyl)Phenyl)-4-Methyl-1,1-Dioxido-1,2,6-Thiadiazinan-2-yl)Acetamido)Adamantan-1-Carboxamide (KR-67607), Prevents BAC-Induced Dry Eye Syndrome
Author
Yoon-Ju Na, Kyoung Jin Choi, Won Hoon Jung, Sung Bum Park, Sein Kang, Jin Hee Ahn and Ki Young Kim*
Year
2020
Source
Int. J. Mol. Sci. 2020, 21, 3729
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